broad_id
string
depmap_id
string
ccle_name
string
screen_id
string
upper_limit
int64
lower_limit
float64
slope
float64
r2
float64
auc
float64
ec50
float64
ic50
float64
name
string
moa
string
target
string
disease.area
string
indication
string
smiles
string
phase
string
passed_str_profiling
bool
row_name
string
BRD-A98990573-003-01-3
ACH-000367
NCIH226_LUNG
HTS002
1
2.478964
0.057529
-0.037068
1.433468
380,001.249781
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000367
BRD-A98990573-003-01-3
ACH-001190
SKMEL2_SKIN
HTS002
1
1.246811
-0.015808
-0.229736
1.150525
149,107,225,833.317
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-001190
BRD-A98990573-003-01-3
ACH-000713
CAOV3_OVARY
HTS002
1
1.346589
0.135358
0.001704
1.168214
0.122368
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000713
BRD-A98990573-003-01-3
ACH-000672
IALM_LUNG
HTS002
1
3.397769
-0.115197
0.097976
1.771578
0.000103
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000672
BRD-A98990573-003-01-3
ACH-000875
NCIH2347_LUNG
HTS002
1
2.050145
0.171866
0.013351
1.467693
0.301243
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000875
BRD-A98990573-003-01-3
ACH-000423
SKMEL3_SKIN
HTS002
1
1.550757
0.143829
0.003124
1.296959
0.02509
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000423
BRD-A98990573-003-01-3
ACH-000553
SQ1_LUNG
HTS002
1
1.429767
0.050656
-0.045753
1.211948
0.134356
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000553
BRD-A98990573-003-01-3
ACH-000834
UMUC1_URINARY_TRACT
HTS002
1
2.420943
-0.386907
0.025175
1.570848
0.02106
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000834
BRD-A98990573-003-01-3
ACH-000252
LS1034_LARGE_INTESTINE
HTS002
1
1.764826
0.318103
0.075741
1.460723
0.016555
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000252
BRD-A98990573-003-01-3
ACH-000123
COV434_OVARY
HTS002
1
1.871036
0.971387
0.042252
1.23525
0.790329
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000123
BRD-A98990573-003-01-3
ACH-000329
CCFSTTG1_CENTRAL_NERVOUS_SYSTEM
HTS002
1
2.043009
-0.033437
-0.174835
1.543977
1.035926
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000329
BRD-A98990573-003-01-3
ACH-000717
COLO680N_OESOPHAGUS
HTS002
1
1.78235
-0.034124
-0.001352
1.389012
0.056457
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000717
BRD-A98990573-003-01-3
ACH-000669
SW900_LUNG
HTS002
1
1.832861
-0.00685
-0.103785
1.426702
105.043676
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000669
BRD-A98990573-003-01-3
ACH-000764
SH10TC_STOMACH
HTS002
1
1.051229
0.112602
-0.402757
1.030866
0.001776
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000764
BRD-A98990573-003-01-3
ACH-000288
BT549_BREAST
HTS002
1
1.701641
0.191987
0.074533
1.347764
0.086103
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000288
BRD-A98990573-003-01-3
ACH-000228
BICR31_UPPER_AERODIGESTIVE_TRACT
HTS002
1
2.25861
0.069242
0.033481
1.551604
2.911644
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000228
BRD-A98990573-003-01-3
ACH-000977
LNCAPCLONEFGC_PROSTATE
HTS002
1
0.971757
0.693095
-0.229357
0.983601
0.033669
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000977
BRD-A98990573-003-01-3
ACH-000397
TEN_ENDOMETRIUM
HTS002
1
2.376421
-0.009003
-0.041521
1.814746
68,925,885,048,248,780
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000397
BRD-A98990573-003-01-3
ACH-000565
RCM1_LARGE_INTESTINE
HTS002
1
1.558587
-0.55099
0.033954
1.278205
0.076446
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000565
BRD-A98990573-003-01-3
ACH-000927
BT474_BREAST
HTS002
1
1.343573
-0.196606
-0.171738
1.231561
4.08948
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000927
BRD-K47832606-001-30-1
ACH-000879
MFE296_ENDOMETRIUM
HTS002
1
0.123092
7.885006
0.523307
0.726373
0.48411
0.501776
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000879
BRD-K47832606-001-30-1
ACH-000320
PSN1_PANCREAS
HTS002
1
0.10514
4.771221
0.972544
0.336463
0.007499
0.007879
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000320
BRD-K47832606-001-30-1
ACH-001145
OC316_OVARY
HTS002
1
0.099077
3.864619
0.803485
0.485618
0.039244
0.041552
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-001145
BRD-K47832606-001-30-1
ACH-000873
KYSE270_OESOPHAGUS
HTS002
1
0.060055
3.816708
0.775195
0.548483
0.094523
0.097745
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000873
BRD-K47832606-001-30-1
ACH-000855
KYSE150_OESOPHAGUS
HTS002
1
0.390028
5.593754
0.711406
0.631609
0.028491
0.037349
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000855
BRD-K47832606-001-30-1
ACH-000913
ESS1_ENDOMETRIUM
HTS002
1
0.27864
2.113099
0.413024
0.647397
0.087092
0.128069
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000913
BRD-K47832606-001-30-1
ACH-000558
A172_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.219398
1.167315
0.603356
0.580288
0.054058
0.088671
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000558
BRD-K47832606-001-30-1
ACH-000593
BC3C_URINARY_TRACT
HTS002
1
0.285356
3.283477
0.629942
0.645974
0.0817
0.105699
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000593
BRD-K47832606-001-30-1
ACH-000488
TE11_OESOPHAGUS
HTS002
1
0.236216
3.808991
0.794521
0.598061
0.060558
0.071628
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000488
BRD-K47832606-001-30-1
ACH-000832
CAL27_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.278338
2.946289
0.812135
0.564635
0.028676
0.037794
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000832
BRD-K47832606-001-30-1
ACH-000781
NCIH2023_LUNG
HTS002
1
0.379814
9.909888
0.441305
0.690942
0.0794
0.091684
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000781
BRD-K47832606-001-30-1
ACH-000833
RH30_SOFT_TISSUE
HTS002
1
0.322819
1.710281
0.592769
0.543245
0.01433
0.026284
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000833
BRD-K47832606-001-30-1
ACH-000137
8MGBA_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.188678
2.328343
0.757438
0.581448
0.066961
0.082072
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000137
BRD-K47832606-001-30-1
ACH-000632
HS944T_SKIN
HTS002
1
0.185653
3.906275
0.661074
0.560786
0.05333
0.060058
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000632
BRD-K47832606-001-30-1
ACH-000319
MPP89_PLEURA
HTS002
1
2.515378
-0.014656
-0.013553
1.771409
0.925875
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000319
BRD-K47832606-001-30-1
ACH-000630
YD8_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.425762
2.865641
0.030134
0.85194
0.819372
1.594198
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000630
BRD-K47832606-001-30-1
ACH-000266
SNU213_PANCREAS
HTS002
1
1.522356
-6.680382
0.191283
1.111944
0.004884
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000266
BRD-K47832606-001-30-1
ACH-000047
GCIY_STOMACH
HTS002
1
0.223612
2.620157
0.775777
0.573586
0.048452
0.060754
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000047
BRD-K47832606-001-30-1
ACH-000273
SF539_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.131052
4.46567
0.760405
0.492328
0.034496
0.036926
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000273
BRD-K47832606-001-30-1
ACH-000682
SNU1066_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.22864
2.817694
0.774301
0.572712
0.046286
0.057498
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000682
BRD-K47832606-001-30-1
ACH-000359
MG63_BONE
HTS002
1
0.293324
2.729806
0.654008
0.750275
0.324131
0.447995
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000359
BRD-K47832606-001-30-1
ACH-000846
FADU_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.101684
0.891676
0.883318
0.492464
0.040847
0.052711
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000846
BRD-K47832606-001-30-1
ACH-000804
NB1_AUTONOMIC_GANGLIA
HTS002
1
0.073301
1.959961
0.972829
0.421177
0.023306
0.025269
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000804
BRD-K47832606-001-30-1
ACH-000609
SF126_CENTRAL_NERVOUS_SYSTEM
HTS002
1
-0.038818
0.519385
0.784649
0.418278
0.030612
0.026508
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000609
BRD-K47832606-001-30-1
ACH-000974
SNGM_ENDOMETRIUM
HTS002
1
0.226438
3.244132
0.466407
0.649378
0.122966
0.148088
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000974
BRD-K47832606-001-30-1
ACH-000987
MEWO_SKIN
HTS002
1
0.149936
1.387641
0.812502
0.592523
0.095506
0.123481
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000987
BRD-K47832606-001-30-1
ACH-000787
LXF289_LUNG
HTS002
1
0.229243
5.140688
0.849299
0.521692
0.024247
0.02732
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000787
BRD-K47832606-001-30-1
ACH-000561
TT_OESOPHAGUS
HTS002
1
0.194131
3.821604
0.732601
0.536222
0.037549
0.042702
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000561
BRD-K47832606-001-30-1
ACH-000212
CAL120_BREAST
HTS002
1
0.169088
1.825458
0.844268
0.639196
0.147939
0.185473
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000212
BRD-K47832606-001-30-1
ACH-000753
JMSU1_URINARY_TRACT
HTS002
1
0.071853
1.297696
0.77363
0.652125
0.265021
0.298676
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000753
BRD-K47832606-001-30-1
ACH-000305
ECGI10_OESOPHAGUS
HTS002
1
0.33356
2.198212
0.786261
0.693634
0.115508
0.190516
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000305
BRD-K47832606-001-30-1
ACH-000138
CFPAC1_PANCREAS
HTS002
1
0.100176
0.899843
0.676359
0.409957
0.016351
0.020963
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000138
BRD-K47832606-001-30-1
ACH-000250
KMRC20_KIDNEY
HTS002
1
0.325036
5.218719
0.656166
0.666281
0.082467
0.100847
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000250
BRD-K47832606-001-30-1
ACH-000856
CAL51_BREAST
HTS002
1
0.242264
5.051557
0.81304
0.571427
0.041337
0.047131
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000856
BRD-K47832606-001-30-1
ACH-000046
ACHN_KIDNEY
HTS002
1
0.032024
2.346294
0.797691
0.441029
0.036839
0.037893
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000046
BRD-K47832606-001-30-1
ACH-000878
HCC15_LUNG
HTS002
1
0.292419
3.746697
0.852231
0.602022
0.042619
0.053889
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000878
BRD-K47832606-001-30-1
ACH-000766
NCIH1648_LUNG
HTS002
1
0.178486
6.801478
0.839077
0.530087
0.038843
0.041448
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000766
BRD-K47832606-001-30-1
ACH-000666
NCIH1355_LUNG
HTS002
1
0.486426
2.745142
0.401085
0.75265
0.093375
0.347363
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000666
BRD-K47832606-001-30-1
ACH-000014
HS294T_SKIN
HTS002
1
0.190261
3.40639
0.653899
0.546061
0.04339
0.04994
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000014
BRD-K47832606-001-30-1
ACH-000701
RMUGS_OVARY
HTS002
1
0.327732
1.554079
0.635325
0.641891
0.056868
0.112887
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000701
BRD-K47832606-001-30-1
ACH-000884
MDAMB435S_SKIN
HTS002
1
1.468327
-2.133493
0.420368
1.246145
0.10014
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000884
BRD-K47832606-001-30-1
ACH-000037
S117_SOFT_TISSUE
HTS002
1
0.24471
2.80327
0.534332
0.647703
0.1082
0.137521
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000037
BRD-K47832606-001-30-1
ACH-000504
SNB75_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.145945
4.673798
0.540869
0.601978
0.108622
0.116947
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000504
BRD-K47832606-001-30-1
ACH-000502
TCCPAN2_PANCREAS
HTS002
1
0.240968
4.698223
0.74694
0.646632
0.109136
0.125534
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000502
BRD-K47832606-001-30-1
ACH-000886
NCIH2009_LUNG
HTS002
1
0.053788
6.749659
0.887671
0.30824
0.008297
0.008438
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000886
BRD-K47832606-001-30-1
ACH-000035
NCIH1650_LUNG
HTS002
1
0.549551
8.693176
0.452271
0.773775
0.076459
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000035
BRD-K47832606-001-30-1
ACH-000661
WM1799_SKIN
HTS002
1
0.172981
0.997392
0.751888
0.459293
0.016976
0.025985
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000661
BRD-K47832606-001-30-1
ACH-000391
MHHES1_BONE
HTS002
1
0.057975
5.871609
0.689743
0.513058
0.066302
0.067708
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000391
BRD-K47832606-001-30-1
ACH-000843
HARA_LUNG
HTS002
1
0.266728
2.027041
0.643432
0.590675
0.044402
0.064677
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000843
BRD-K47832606-001-30-1
ACH-000711
JIMT1_BREAST
HTS002
1
0.258613
3.917281
0.331083
0.668526
0.130536
0.157205
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000711
BRD-K47832606-001-30-1
ACH-000232
U251MG_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.111125
1.786807
0.673534
0.508229
0.046588
0.053625
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000232
BRD-K47832606-001-30-1
ACH-000060
PANC1005_PANCREAS
HTS002
1
0.365577
5.680825
0.614259
0.653408
0.049844
0.062812
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000060
BRD-K47832606-001-30-1
ACH-000322
HT144_SKIN
HTS002
1
0.156055
4.765827
0.456102
0.617693
0.123272
0.133339
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000322
BRD-K47832606-001-30-1
ACH-000736
SNU601_STOMACH
HTS002
1
0.064045
2.857174
0.893413
0.338135
0.010464
0.010978
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000736
BRD-K47832606-001-30-1
ACH-000809
KYSE410_OESOPHAGUS
HTS002
1
0.249972
1.284933
0.829526
0.563619
0.035185
0.060339
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000809
BRD-K47832606-001-30-1
ACH-000747
NCIH1703_LUNG
HTS002
1
0.104899
1.18601
0.90381
0.676512
0.303697
0.370394
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000747
BRD-K47832606-001-30-1
ACH-000364
U2OS_BONE
HTS002
1
1.435834
-6.467609
0.29223
1.137719
0.013101
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000364
BRD-K47832606-001-30-1
ACH-000679
OE19_OESOPHAGUS
HTS002
1
0.23987
4.833581
0.682862
0.658406
0.127667
0.146147
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000679
BRD-K47832606-001-30-1
ACH-000985
LS411N_LARGE_INTESTINE
HTS002
1
0.148856
3.086933
0.699415
0.539835
0.052662
0.05905
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000985
BRD-K47832606-001-30-1
ACH-000441
SH4_SKIN
HTS002
1
0.502221
5.618827
0.659641
0.770076
0.113072
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000441
BRD-K47832606-001-30-1
ACH-001113
LC1SQSF_LUNG
HTS002
1
0.482338
3.09893
0.214854
0.764082
0.12004
0.353063
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-001113
BRD-K47832606-001-30-1
ACH-000620
JHH1_LIVER
HTS002
1
0.655783
9.945614
0.358919
0.827884
0.078108
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000620
BRD-K47832606-001-30-1
ACH-000853
NCIH661_LUNG
HTS002
1
0.52168
2.862689
0.48102
0.768694
0.091619
null
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000853
BRD-K47832606-001-30-1
ACH-000102
GMS10_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.250206
1.810383
0.68131
0.579092
0.04306
0.063176
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000102
BRD-K47832606-001-30-1
ACH-000648
NCIH28_PLEURA
HTS002
1
0.28697
7.031266
0.539409
0.666134
0.10633
0.120048
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000648
BRD-K47832606-001-30-1
null
null
HTS002
1
0.131836
1.959351
0.906137
0.401642
0.012437
0.01454
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
false
ACH-000925_FAILED_STR
BRD-K47832606-001-30-1
ACH-001239
WM2664_SKIN
HTS002
1
0.163677
2.237879
0.855226
0.565935
0.064959
0.077552
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-001239
BRD-K47832606-001-30-1
ACH-001321
TT_THYROID
HTS002
1
0.384921
3.278042
0.722054
0.835351
0.744516
1.165452
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-001321
BRD-K47832606-001-30-1
ACH-000279
EWS502_BONE
HTS002
1
0.062731
1.855873
0.74678
0.431616
0.027802
0.029884
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000279
BRD-K47832606-001-30-1
ACH-000172
TM87_SOFT_TISSUE
HTS002
1
0.110156
3.392582
0.895632
0.5249
0.056216
0.060494
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000172
BRD-K47832606-001-30-1
ACH-001128
MON_SOFT_TISSUE
HTS002
1
0.125018
9.151695
0.585093
0.569529
0.08445
0.087147
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-001128
BRD-K47832606-001-30-1
ACH-000437
SW1088_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.109291
1.89719
0.694857
0.393217
0.013438
0.015304
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000437
BRD-K47832606-001-30-1
ACH-000735
PECAPJ49_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.09273
1.218993
0.882721
0.39397
0.015064
0.017824
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000735
BRD-K47832606-001-30-1
ACH-000643
HDQP1_BREAST
HTS002
1
0.379726
7.466043
0.719555
0.696771
0.087041
0.105343
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000643
BRD-K47832606-001-30-1
ACH-000207
DETROIT562_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.266922
3.327026
0.572965
0.590454
0.044212
0.055612
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000207
BRD-K47832606-001-30-1
ACH-000456
BCPAP_THYROID
HTS002
1
0.054028
0.735584
0.795512
0.506728
0.062682
0.073225
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000456
BRD-K47832606-001-30-1
ACH-000260
SKNAS_AUTONOMIC_GANGLIA
HTS002
1
0.219911
5.482424
0.412103
0.558627
0.041256
0.045855
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000260
BRD-K47832606-001-30-1
ACH-000019
MCF7_BREAST
HTS002
1
0.331773
1.034922
0.695635
0.706686
0.142477
0.408183
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000019
BRD-K47832606-001-30-1
ACH-000582
COLO741_SKIN
HTS002
1
0.26895
1.045834
0.580407
0.71155
0.220731
0.461781
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000582
BRD-K47832606-001-30-1
ACH-000990
HEC108_ENDOMETRIUM
HTS002
1
0.346441
3.549785
0.620228
0.650627
0.055859
0.077898
floxuridine
DNA synthesis inhibitor
TYMS
oncology
colorectal cancer
OC[C@H]1OC(C[C@H]1O)n1cc(F)c(=O)[nH]c1=O, OC[C@H]1O[C@H](C[C@@H]1O)n1cc(F)c(=O)[nH]c1=O
Launched
true
ACH-000990